Birger Brodin Larsen
Professor
CNS Drug Delivery and Barrier Modelling
Universitetsparken 2
2100 København Ø
- 2020
- Udgivet
The Pyrazolo[3,4-d]pyrimidine Derivative, SCO-201, Reverses Multidrug Resistance Mediated by ABCG2/BCRP
Ambjørner, S. E. B., Wiese, M., Köhler, S. C., Svindt, J., Lund, X. L., Gajhede, Michael, Saaby, Lasse, Larsen, Birger Brodin, Rump, S., Weigt, H., Brünner, N. & Stenvang, Jan, 4 mar. 2020, I: Cells. 9, 3, 22 s., 613.Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
- Udgivet
Conjugation of Therapeutic PSD-95 Inhibitors to the Cell-Penetrating Peptide Tat Affects Blood-Brain Barrier Adherence, Uptake, and Permeation
Kristensen, Mie, Kucharz, Krzysztof, Alves Fernandes, Eduardo Felipe, Strømgaard, Kristian, Schallburg Nielsen, M., Cederberg Helms, H. C., Bach, Anders, Ulrikkaholm Tofte-Hansen, M., Aldana, Blanca, Lauritzen, Martin & Larsen, Birger Brodin, 2020, I: Pharmaceutics. 12, 7, 24 s., 661.Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
- Udgivet
Drug Delivery Strategies to Overcome the Blood-Brain Barrier (BBB)
Helms, H. C. C., Kristensen, Mie, Saaby, Lasse, Fricker, G. & Larsen, Birger Brodin, 2020, Handbook of Experimental Pharmacology. Springer, Bind 273. s. 151-183Publikation: Bidrag til bog/antologi/rapport › Bidrag til bog/antologi › Formidling
- 2019
- Udgivet
miRNA-27a-3p and miRNA-222-3p as Novel Modulators of Phosphodiesterase 3a (PDE3A) in Cerebral Microvascular Endothelial Cells
Yasmeen, S., Kaur, S., Mirza, A. H., Larsen, Birger Brodin, Pociot, Flemming & Kruuse, Christina Rostrup, aug. 2019, I: Molecular Neurobiology. 56, 8, s. 5304–5314Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
- Udgivet
Effects of oxygen-glucose deprivation (OGD) on barrier properties and mRNA transcript levels of selected marker proteins in brain endothelial cells/astrocyte co-cultures
Tornabene, E., Helms, H. C. C., Pedersen, Stine Helene Falsig & Larsen, Birger Brodin, 2019, I: PLoS ONE. 14, 8, 20 s., e0221103.Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
- Udgivet
Evaluating the involvement of cerebral microvascular endothelial Na+/K+-ATPase and Na+-K+-2Cl- co-transporter in electrolyte fluxes in an in vitro blood-brain barrier model of dehydration
Lykke, K., Assentoft, M., Hørlyck, S., Helms, H. C. C., Stoica, A., Toft-Bertelsen, Trine Lisberg, Tritsaris, Katerina, Vilhardt, Frederik, Larsen, Birger Brodin & MacAulay, Nanna, 2019, I: Journal of Cerebral Blood Flow and Metabolism. 39, 3, s. 497-512Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
- Udgivet
Two-photon fluorescence imaging: a platform to investigate cell-penetrating peptides and liposome-based nanocarriers for drug delivery across the heterogeneous BBB in vivo
Kucharz, K., Kristensen, K., Kristensen, Mie, Lund, M., Andresen, T., Larsen, Birger Brodin & Lauritzen, M., 2019, I: Journal of Cerebral Blood Flow and Metabolism. 39, s. 60 1 s.Publikation: Bidrag til tidsskrift › Konferenceabstrakt i tidsskrift › Forskning › fagfællebedømt
- 2018
- Udgivet
Validation of reference genes for normalization of real-time quantitative PCR studies of gene expression in brain capillary endothelial cells cultured in vitro
Hersom, M., Goldeman, C., Pretzer, N. & Larsen, Birger Brodin, dec. 2018, I: Molecular and Cellular Neuroscience. 93, s. 27-35 9 s.Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
- Udgivet
The iP-gp cell model is an improved tool for predicting the in vivo relevance of P-gp mediated efflux at the blood-brain barrier
Ozgür, Burak, Saaby, Lasse, Eneberg, E., Langthaler, K., Jacobsen, A., Janfelt, Christian, Badolo, L., Montanari, D. & Larsen, Birger Brodin, 22 jun. 2018.Publikation: Konferencebidrag › Poster › Forskning › fagfællebedømt
- Udgivet
Characterization of the IPEC-J2 MDR1 (iP-gp) cell line as a tool for identification of P-gp substrates
Ozgür, Burak, Saaby, Lasse, Langthaler, K. & Larsen, Birger Brodin, 2018, I: European Journal of Pharmaceutical Sciences. 112, s. 112-121 10 s.Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
- Udgivet
Data demonstrating the challenges of determining the kinetic parameters of P-gp mediated transport of low-water soluble substrates
Ozgür, Burak, Saaby, Lasse, Langthaler, K. & Larsen, Birger Brodin, 2018, I: Data in Brief. 16, s. 655-659 5 s.Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
- Udgivet
Stimulation-induced increases in cerebral blood flow and local capillary vasoconstriction depend on conducted vascular responses
Cai, Changsi, Fordsmann, J. C., Jensen, S. H., Gesslein, B., wbh615, wbh615, Hald, B. O., Zambach, S. A., Larsen, Birger Brodin & Lauritzen, Martin, 2018, I: Proceedings of the National Academy of Sciences of the United States of America. 115, 25, s. E5796-E5804 9 s.Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
- Udgivet
The insulin receptor is expressed and functional in cultured blood-brain barrier endothelial cells, but does not mediate insulin entry from blood-to-brain
Hersom, M., Helms, H. C., Schmalz, C., Pedersen, T. Å., Buckley, S. T. & Larsen, Birger Brodin, 2018, I: American Journal of Physiology: Endocrinology and Metabolism. 315, 4, s. E531-E542Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
- 2017
- Udgivet
Substrate-Dependent Inhibition of P-glycoprotein Mediated Efflux Transport of Digoxin
Saaby, L., Ozgür, Burak & Larsen, Birger Brodin, 14 nov. 2017, s. T7089.Publikation: Konferencebidrag › Konferenceabstrakt til konference › Forskning › fagfællebedømt
- Udgivet
Current research into brain barriers and the delivery of therapeutics for neurological diseases: a report on CNS barrier congress London, UK, 2017
Greenwood, J., Hammarlund-Udenaes, M., Jones, H. C., Stitt, A. W., Vandenbrouke, R. E., Romero, I. A., Campbell, M., Fricker, G., Larsen, Birger Brodin, Manninga, H., Gaillard, P. J., Schwaninger, M., Webster, C., Wicher, K. B. & Khrestchatisky, M., 7 nov. 2017, I: Fluids and Barriers of the CNS. 14, 11 s., 31.Publikation: Bidrag til tidsskrift › Review › Forskning › fagfællebedømt
- Udgivet
Development and Characterization of a Brain Endothelial Cell Phenotype using Human Induced Pluripotent Stem Cells
Goldeman, C., Saaby, L., Holst, B., Hall, Vanessa Jane, Hyttel, P. & Larsen, Birger Brodin, 2 nov. 2017.Publikation: Konferencebidrag › Poster › Forskning › fagfællebedømt
- Udgivet
A Critical View on In Vitro Analysis of P-glycoprotein (P-gp) Transport Kinetics
Saaby, Lasse & Larsen, Birger Brodin, sep. 2017, I: Journal of Pharmaceutical Sciences. 106, 9, s. 2257-2264 8 s.Publikation: Bidrag til tidsskrift › Review › Forskning › fagfællebedømt
- Udgivet
Routes for drug translocation across the blood-brain barrier: Exploiting peptides as delivery vectors
Kristensen, Mie & Larsen, Birger Brodin, sep. 2017, I: Journal of Pharmaceutical Sciences. 106, 9, s. 2326-2334Publikation: Bidrag til tidsskrift › Review › Forskning › fagfællebedømt
- Udgivet
iP-gp , a novel cell line with tight barrier function and expression of human P-glycoprotein (ABCB1) for drug screening
Larsen, Birger Brodin, Ozgür, Burak & Saaby, Lasse, 23 maj 2017.Publikation: Konferencebidrag › Konferenceabstrakt til konference › Forskning › fagfællebedømt
- Udgivet
Bidirectional apical-basal traffic of the cation-independent mannose-6-phosphate receptor in brain endothelial cells
Siupka, P., Hersom, M. N., Lykke-Hartmann, K., Johnsen, K. B., Thomsen, L. B., Andresen, T. L., Moos, T., Abbott, N. J. & Larsen, Birger Brodin, 1 jan. 2017, I: Journal of Cerebral Blood Flow and Metabolism. 37, 7, s. 2598-2613Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
- Udgivet
Characterization of the L-glutamate clearance pathways across the blood-brain barrier and the effect of astrocytes in an in vitro blood-brain barrier model
Helms, H. C., Aldana, Blanca, Groth, S., Jensen, M. M., Waagepetersen, Helle S., Nielsen, C. U. & Larsen, Birger Brodin, 2017, I: Journal of Cerebral Blood Flow and Metabolism. 37, 12, s. 3744–3758Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › fagfællebedømt
- Udgivet
Glutamate Transporters in the Blood-Brain Barrier
Helms, H. C. C., Nielsen, C. U., Waagepetersen, Helle S. & Larsen, Birger Brodin, 2017, Glial Amino Acid Transporters. Bind 16. s. 297-314 18 s. (Advances in Neurobiology).Publikation: Bidrag til bog/antologi/rapport › Bidrag til bog/antologi › Forskning › fagfællebedømt
- 2016
- Udgivet
Initial Attempts of Development and Characterization of an In Vitro Blood Brain Barrier Model Derived from Human Pluripotent Stem Cells
Goldeman, C., Saaby, L., Hall, Vanessa Jane, Hyttel, P. & Larsen, Birger Brodin, 8 dec. 2016. 1 s.Publikation: Konferencebidrag › Poster › Forskning › fagfællebedømt
- Udgivet
Down-regulation of selected Blood-brain Barrier Specific Genes from Capillaries to Bovine In Vitro Models
Goldeman, C., Saaby, L. & Larsen, Birger Brodin, 14 sep. 2016. 1 s.Publikation: Konferencebidrag › Poster › Forskning › fagfællebedømt
- Udgivet
The insulin receptor is expressed and functional in blood-brain barrier endothelial cells, but does not mediate insulin entry from blood-to-brain
Hersom, M. N. S., Helms, H. C. C., Pedersen, T., Buckley, S. & Larsen, Birger Brodin, 14 sep. 2016.Publikation: Konferencebidrag › Konferenceabstrakt til konference › Forskning
ID: 1299175
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Design of prodrugs targeting the intestinal di/tri‐peptide transporter hPEPT1 (SLC15A1
Publikation: Konferencebidrag › Konferenceabstrakt til konference › Forskning › fagfællebedømt
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A bovine in vitro blood-brain barrier model under oxygenglucose deprivation (OGD) condition
Publikation: Konferencebidrag › Poster › Forskning
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